Name | Synonyms | Targets | Target Pathway | PubCHEM | Datatset | Sample size | Screening site |
---|---|---|---|---|---|---|---|
A-443654 | KIN001-139 | AKT1, AKT2, AKT3 | PI3K/MTOR signaling | 10172943 | GDSC1 | 397 | MGH |
AKT inhibitor VIII | Akti-1/2, KIN001-102 | AKT1, AKT2, AKT3 | PI3K/MTOR signaling | 10196499 | GDSC1 | 877 | MGH |
AKT inhibitor VIII | Akti-1/2, KIN001-102 | AKT1, AKT2, AKT3 | PI3K/MTOR signaling | 10196499 | GDSC1 | 913 | MGH |
AZD5363 | AKT1, AKT2, AKT3, ROCK2 | Other, kinases | 25227436, 42602260 | GDSC2 | 958 | SANGER | |
Afuresertib | GSK2110183, GSK2110183C | AKT1, AKT2, AKT3 | PI3K/MTOR signaling | 46843057 | GDSC2 | 957 | SANGER |
BAY AKT1 | AKT1, AKT2, AKT3 | Apoptosis regulation | GDSC1 | 835 | SANGER | ||
GSK2110183B | AKT1, AKT2, AKT3 | PI3K/MTOR signaling | GDSC2 | 717 | SANGER | ||
GSK690693 | GSK 690693, GSK-690693 | AKT1, AKT2, AKT3 | PI3K/MTOR signaling | 16725726 | GDSC1 | 910 | MGH |
Ipatasertib | GDC0068, GDC 0068, GDC-0068 | AKT1, AKT, AKT3 | PI3K/MTOR signaling | 24788740 | GDSC2 | 958 | SANGER |
Uprosertib | GSK2141795, GSK2141795C, GSK-2141795 | AKT1, AKT2, AKT3 | PI3K/MTOR signaling | 51042438 | GDSC2 | 898 | SANGER |
Uprosertib | GSK2141795, GSK2141795C, GSK-2141795 | AKT1, AKT2, AKT3 | PI3K/MTOR signaling | 51042438 | GDSC2 | 736 | SANGER |
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