Search Results for: egfr

Name Synonyms Targets Target Pathway PubCHEM Datatset Sample size Screening site
AST-1306 EGFR, ERBB4 RTK signaling GDSC1 903 MGH
AZD3759 EGFR EGFR signaling 78209992 GDSC2 966 SANGER
AZD8931 SN0216062465 EGFR, ERBB2, ERBB3 RTK signaling GDSC1 913 SANGER
Afatinib BIBW2992, Tovok, Gilotrif EGFR, ERBB2 EGFR signaling 10184653 GDSC1 929 SANGER
Afatinib BIBW2992, Tovok, Gilotrif EGFR, ERBB2 EGFR signaling 10184653 GDSC1 903 SANGER
Afatinib BIBW2992, Tovok, Gilotrif EGFR, ERBB2 EGFR signaling 10184653 GDSC2 966 SANGER
Axitinib AG-13736, Inlyta PDGFR, KIT, VEGFR RTK signaling 6450551 GDSC1 927 SANGER
Axitinib AG-13736, Inlyta PDGFR, KIT, VEGFR RTK signaling 6450551 GDSC2 961 SANGER
BIBF-1120 VEGFR, PDGFR, FGFR RTK signaling GDSC1 918 MGH
Brivanib, BMS-540215 VEGFR, PDGFR RTK signaling GDSC1 918 MGH
CI-1033 EGFR, ERBB2, ERBB4 RTK signaling GDSC1 916 MGH
CUDC-101 CUDC 101 HDAC1-10, EGFR, ERBB2 Other 24756910 GDSC1 893 MGH
Cabozantinib BMS-907351, XL-184, Cometriq VEGFR, MET, RET, KIT, FLT1, FLT3, FLT4, TIE2,AXL RTK signaling 25102847 GDSC1 911 MGH
Cediranib AZD2171, AZD 2171, AZD-2171, Recentin VEGFR, FLT1, FLT2, FLT3, FLT4, KIT, PDGFRB RTK signaling 9933475 GDSC2 958 SANGER
Cetuximab Erbitux, IMC-C225, C225, IMC-225, L01XC06 EGFR EGFR signaling 85668777 GDSC1 862 SANGER
Erlotinib Tarceva, RG-1415, CP-358774, OSI-774, Ro-508231, R-1415 EGFR EGFR signaling 176870 GDSC1 393 MGH
Erlotinib Tarceva, RG-1415, CP-358774, OSI-774, Ro-508231, R-1415 EGFR EGFR signaling 176870 GDSC2 955 SANGER
Foretinib GSK1363089, XL-880, EXEL-2880, GSK089 MET, KDR, TIE2, VEGFR3/FLT4, RON, PDGFR, FGFR1, EGFR RTK signaling 42642645 GDSC1 909 MGH
Foretinib GSK1363089, XL-880, EXEL-2880, GSK089 MET, KDR, TIE2, VEGFR3/FLT4, RON, PDGFR, FGFR1, EGFR RTK signaling 42642645 GDSC2 953 SANGER
Gefitinib ZD-1839, Iressa EGFR EGFR signaling 123631 GDSC1 927 SANGER
Gefitinib ZD-1839, Iressa EGFR EGFR signaling 123631 GDSC2 958 SANGER
Lapatinib Tykerb, Tyverb EGFR, ERBB2 RTK signaling 208908 GDSC1 395 MGH
Lapatinib Tykerb, Tyverb EGFR, ERBB2 EGFR signaling 208908 GDSC2 966 SANGER
Linifanib ABT-869, ABT 869 VEGFR1, VEGFR2, VEGFR3, CSF1R, FLT3, KIT RTK signaling 11485656 GDSC1 914 MGH
Motesanib AMG-706, AMG 706, AMG706 VEGFR, RET, KIT, PDGFR RTK signaling 11667893 GDSC1 927 SANGER
Motesanib AMG-706, AMG 706, AMG706 VEGFR, RET, KIT, PDGFR RTK signaling 11667893 GDSC2 949 SANGER
OSI-930 OSI 930 OSI930 KIT, VEGFR2 RTK signaling 9868037 GDSC1 913 MGH
Osimertinib AZD9291, AZD 9291, AZD-9291, Tagrisso, Mereletinib EGFR EGFR signaling 71496458 GDSC2 957 SANGER
PF-00299804 EGFR, ERBB2, ERBB4 RTK signaling GDSC1 909 MGH
Pelitinib EKB-569, EKB 569 EGFR EGFR signaling 6445562 GDSC1 913 MGH
Ponatinib AP24534, AP-24534, KIN001-192, Iclusig ABL, PDGFRA, VEGFR2, FGFR1, SRC, TIE2, FLT3 Other, kinases 24826799 GDSC1 877 MGH
Sapitinib AZD8931 EGFR, ERBB2, ERBB3 EGFR signaling 11488320 GDSC2 966 SANGER
Sorafenib Nexavar, 284461-73-0, BAY 43-9006 PDGFR, KIT, VEGFR, RAF RTK signaling 216239 GDSC1 396 MGH
Sorafenib Nexavar, 284461-73-0, BAY 43-9006 PDGFR, KIT, VEGFR, RAF Other, kinases 216239 GDSC2 958 SANGER
Sunitinib Sutent, Sunitinib Malate, SU-11248 PDGFR, KIT, VEGFR, FLT3, RET, CSF1R RTK signaling 5329102 GDSC1 396 MGH
Tivozanib AV-951, AV 951, KRN-951, KIL8951, ASP-4130 VEGFR1, VEGFR2, VEGFR3, PDGFR, KIT RTK signaling 9911830 GDSC1 912 MGH
Feature Name Feature Type
EGFR_mut coding variant

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