AST-1306 |
|
EGFR, ERBB4 |
RTK signaling |
|
GDSC1 |
903 |
MGH |
AZD3759 |
|
EGFR |
EGFR signaling |
78209992 |
GDSC2 |
966 |
SANGER |
AZD8931 |
SN0216062465 |
EGFR, ERBB2, ERBB3 |
RTK signaling |
|
GDSC1 |
913 |
SANGER |
Afatinib |
BIBW2992, Tovok, Gilotrif |
EGFR, ERBB2 |
EGFR signaling |
10184653 |
GDSC1 |
929 |
SANGER |
Afatinib |
BIBW2992, Tovok, Gilotrif |
EGFR, ERBB2 |
EGFR signaling |
10184653 |
GDSC1 |
903 |
SANGER |
Afatinib |
BIBW2992, Tovok, Gilotrif |
EGFR, ERBB2 |
EGFR signaling |
10184653 |
GDSC2 |
966 |
SANGER |
Axitinib |
AG-13736, Inlyta |
PDGFR, KIT, VEGFR |
RTK signaling |
6450551 |
GDSC1 |
927 |
SANGER |
Axitinib |
AG-13736, Inlyta |
PDGFR, KIT, VEGFR |
RTK signaling |
6450551 |
GDSC2 |
961 |
SANGER |
BIBF-1120 |
|
VEGFR, PDGFR, FGFR |
RTK signaling |
|
GDSC1 |
918 |
MGH |
Brivanib, BMS-540215 |
|
VEGFR, PDGFR |
RTK signaling |
|
GDSC1 |
918 |
MGH |
CI-1033 |
|
EGFR, ERBB2, ERBB4 |
RTK signaling |
|
GDSC1 |
916 |
MGH |
CUDC-101 |
CUDC 101 |
HDAC1-10, EGFR, ERBB2 |
Other |
24756910 |
GDSC1 |
893 |
MGH |
Cabozantinib |
BMS-907351, XL-184, Cometriq |
VEGFR, MET, RET, KIT, FLT1, FLT3, FLT4, TIE2,AXL |
RTK signaling |
25102847 |
GDSC1 |
911 |
MGH |
Cediranib |
AZD2171, AZD 2171, AZD-2171, Recentin |
VEGFR, FLT1, FLT2, FLT3, FLT4, KIT, PDGFRB |
RTK signaling |
9933475 |
GDSC2 |
958 |
SANGER |
Cetuximab |
Erbitux, IMC-C225, C225, IMC-225, L01XC06 |
EGFR |
EGFR signaling |
85668777 |
GDSC1 |
862 |
SANGER |
Erlotinib |
Tarceva, RG-1415, CP-358774, OSI-774, Ro-508231, R-1415 |
EGFR |
EGFR signaling |
176870 |
GDSC1 |
393 |
MGH |
Erlotinib |
Tarceva, RG-1415, CP-358774, OSI-774, Ro-508231, R-1415 |
EGFR |
EGFR signaling |
176870 |
GDSC2 |
955 |
SANGER |
Foretinib |
GSK1363089, XL-880, EXEL-2880, GSK089 |
MET, KDR, TIE2, VEGFR3/FLT4, RON, PDGFR, FGFR1, EGFR |
RTK signaling |
42642645 |
GDSC1 |
909 |
MGH |
Foretinib |
GSK1363089, XL-880, EXEL-2880, GSK089 |
MET, KDR, TIE2, VEGFR3/FLT4, RON, PDGFR, FGFR1, EGFR |
RTK signaling |
42642645 |
GDSC2 |
953 |
SANGER |
Gefitinib |
ZD-1839, Iressa |
EGFR |
EGFR signaling |
123631 |
GDSC1 |
927 |
SANGER |
Gefitinib |
ZD-1839, Iressa |
EGFR |
EGFR signaling |
123631 |
GDSC2 |
958 |
SANGER |
Lapatinib |
Tykerb, Tyverb |
EGFR, ERBB2 |
RTK signaling |
208908 |
GDSC1 |
395 |
MGH |
Lapatinib |
Tykerb, Tyverb |
EGFR, ERBB2 |
EGFR signaling |
208908 |
GDSC2 |
966 |
SANGER |
Linifanib |
ABT-869, ABT 869 |
VEGFR1, VEGFR2, VEGFR3, CSF1R, FLT3, KIT |
RTK signaling |
11485656 |
GDSC1 |
914 |
MGH |
Motesanib |
AMG-706, AMG 706, AMG706 |
VEGFR, RET, KIT, PDGFR |
RTK signaling |
11667893 |
GDSC1 |
927 |
SANGER |
Motesanib |
AMG-706, AMG 706, AMG706 |
VEGFR, RET, KIT, PDGFR |
RTK signaling |
11667893 |
GDSC2 |
949 |
SANGER |
OSI-930 |
OSI 930 OSI930 |
KIT, VEGFR2 |
RTK signaling |
9868037 |
GDSC1 |
913 |
MGH |
Osimertinib |
AZD9291, AZD 9291, AZD-9291, Tagrisso, Mereletinib |
EGFR |
EGFR signaling |
71496458 |
GDSC2 |
957 |
SANGER |
PF-00299804 |
|
EGFR, ERBB2, ERBB4 |
RTK signaling |
|
GDSC1 |
909 |
MGH |
Pelitinib |
EKB-569, EKB 569 |
EGFR |
EGFR signaling |
6445562 |
GDSC1 |
913 |
MGH |
Ponatinib |
AP24534, AP-24534, KIN001-192, Iclusig |
ABL, PDGFRA, VEGFR2, FGFR1, SRC, TIE2, FLT3 |
Other, kinases |
24826799 |
GDSC1 |
877 |
MGH |
Sapitinib |
AZD8931 |
EGFR, ERBB2, ERBB3 |
EGFR signaling |
11488320 |
GDSC2 |
966 |
SANGER |
Sorafenib |
Nexavar, 284461-73-0, BAY 43-9006 |
PDGFR, KIT, VEGFR, RAF |
RTK signaling |
216239 |
GDSC1 |
396 |
MGH |
Sorafenib |
Nexavar, 284461-73-0, BAY 43-9006 |
PDGFR, KIT, VEGFR, RAF |
Other, kinases |
216239 |
GDSC2 |
958 |
SANGER |
Sunitinib |
Sutent, Sunitinib Malate, SU-11248 |
PDGFR, KIT, VEGFR, FLT3, RET, CSF1R |
RTK signaling |
5329102 |
GDSC1 |
396 |
MGH |
Tivozanib |
AV-951, AV 951, KRN-951, KIL8951, ASP-4130 |
VEGFR1, VEGFR2, VEGFR3, PDGFR, KIT |
RTK signaling |
9911830 |
GDSC1 |
912 |
MGH |