Name | Synonyms | Targets | Target Pathway | PubCHEM | Datatset | Sample size | Screening site |
---|---|---|---|---|---|---|---|
CPI-637 | EP300 | Chromatin histone methylation | GDSC2 | 741 | SANGER | ||
I-CBP112 | EP300, CBP | Chromatin histone acetylation | GDSC1 | 830 | SANGER | ||
SGC-CBP30 | 8-(3-chloro-4-methoxy-phenethyl)-4-(3,5-dimethyl-isoxazol-4-yl)-9-(2-(morpholin-4-yl)-propyl)-7,9-diaza-bicyclo[4.3.0]nona-1(6),2,4,7-tetraene | EP300, CBP | Chromatin histone acetylation | GDSC2 | 716 | SANGER |
Feature Name | Feature Type |
---|---|
EP300_mut | coding variant |
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