Search Results for: met

Name Synonyms Targets Target Pathway PubCHEM Datatset Sample size Screening site
5-Fluorouracil 5-FU Antimetabolite (DNA & RNA) Other 3385 GDSC1 907 MGH
5-Fluorouracil 5-FU Antimetabolite (DNA & RNA) Other 3385 GDSC2 968 SANGER
5-azacytidine DNA methyltransferases Other GDSC2 740 SANGER
AZD6094 SN1042487586 MET RTK signaling GDSC1 919 SANGER
Ara-G 9-??-D-Arabinofuranosyl guanine Anti-metabolite Other GDSC1 906 MGH
BDILV000379a 4-(4-(1-methyl-1H-pyrazol-4-yl)-1-(2-(1-methyl-1H-pyrazol-4-yl)ethyl)-4,5-dihydro-1H-imidazol-5-yl)benzonitrile BAZ2A, BAZ2B Chromatin histone acetylation GDSC2 717 SANGER
BDOCA000347a 4-bromo-N-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methylbenzenesulfonamide BRPF1, BRPF2, BRPF3 Chromatin histone acetylation GDSC2 717 SANGER
Bromosporine ethyl N-[6-(3-methanesulfonamido-4-methylphenyl)-3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-8-yl]carbamate CECR2, BRD2, BRD4, BRD9 Chromatin other GDSC2 716 SANGER
CPI-613 Metabo, Mitochondria Other GDSC1 909 MGH
Cabozantinib BMS-907351, XL-184, Cometriq VEGFR, MET, RET, KIT, FLT1, FLT3, FLT4, TIE2,AXL RTK signaling 25102847 GDSC1 911 MGH
Crizotinib Xalkori, PF2341066, PF-2341066, PF 2341066 MET, ALK, ROS1 RTK signaling 11626560 GDSC1 405 MGH
Crizotinib Xalkori, PF2341066, PF-2341066, PF 2341066 MET, ALK, ROS1 RTK signaling 11626560 GDSC2 966 SANGER
Cytarabine Ara-Cytidine, Arabinosyl Cytosine, U-19920 Antimetabolite Other 6253 GDSC1 923 SANGER
Cytarabine Ara-Cytidine, Arabinosyl Cytosine, U-19920 Antimetabolite Other 6253 GDSC2 743 SANGER
DMOG Dimethyloxalylglcine HIF-PH Metabolism 560326 GDSC1 876 MGH
EPZ5676 EPZ-5676, Pinometostat DOT1L Chromatin histone methylation 57345410 GDSC2 962 SANGER
FY026 [(para-cymene)osmium(N,N-dimethylphenlyazopyridine)(iodide)]hexafluorophophate Unclassified GDSC1 915 SANGER
Fludarabine Fludara Antimetabolite DNA replication GDSC2 717 SANGER
Foretinib GSK1363089, XL-880, EXEL-2880, GSK089 MET, KDR, TIE2, VEGFR3/FLT4, RON, PDGFR, FGFR1, EGFR RTK signaling 42642645 GDSC1 909 MGH
Foretinib GSK1363089, XL-880, EXEL-2880, GSK089 MET, KDR, TIE2, VEGFR3/FLT4, RON, PDGFR, FGFR1, EGFR RTK signaling 42642645 GDSC2 953 SANGER
GSK2801 1-(7-(2-methylsulfonyl-phenyl)-4-propoxy-1-aza-bicyclo[4.3.0]nona-2,4,6,8-tetraen-9-yl)-ethanone Chromatin other GDSC2 717 SANGER
Gemcitabine Gemzar, LY-188011 Pyrimidine antimetabolite DNA replication 60750 GDSC1 859 MGH
Gemcitabine Pyrimidine antimetabolite DNA replication GDSC1 920 SANGER
Gemcitabine Gemzar, LY-188011 Pyrimidine antimetabolite DNA replication 60750 GDSC2 960 SANGER
JNJ38877605 MET RTK signaling GDSC1 917 MGH
MetAP2 Inhibitor, A832234 MetAP2 Other GDSC1 903 MGH
Methotrexate Abitrexate, Amethopterin, Rheumatrex, Trexall, Folex Antimetabolite DNA replication 126941 GDSC1 933 SANGER
Methotrexate Abitrexate, Amethopterin, Rheumatrex, Trexall, Folex Antimetabolite DNA replication 126941 GDSC2 881 SANGER
N-acetyl cysteine NAC Metabolism Metabolism None GDSC2 735 SANGER
N23918-95-7 JMJ histone demethylase Chromatin histone methylation GDSC1 913 SANGER
N24798-49-A1 JMJ histone demethylase Chromatin histone methylation GDSC1 908 SANGER
PHA-665752 PHA665752, PHA 665752 MET RTK signaling 10461815 GDSC1 405 MGH
PRIMA-1MET Prima 1MET, APR-246 TP53 activation p53 pathway 52918385 GDSC2 894 SANGER
Pemetrexed TYMS DNA replication GDSC1 899 MGH
Pyrimethamine Daraprim, Chloridine Dihydrofolate reductase (DHFR) Other 4993 GDSC1 398 MGH
Refametinib RDEA119, BAY-86-9766, BAY 869766 MEK1, MEK2 ERK MAPK signaling 44182295 GDSC1 913 SANGER
Refametinib RDEA119, BAY-86-9766, BAY 869766 MEK1, MEK2 ERK MAPK signaling 44182295 GDSC1 861 SANGER
Refametinib RDEA119, BAY-86-9766, BAY 869766 MEK1, MEK2 ERK MAPK signaling 44182295 GDSC2 947 SANGER
SGC-CBP30 8-(3-chloro-4-methoxy-phenethyl)-4-(3,5-dimethyl-isoxazol-4-yl)-9-(2-(morpholin-4-yl)-propyl)-7,9-diaza-bicyclo[4.3.0]nona-1(6),2,4,7-tetraene EP300, CBP Chromatin histone acetylation GDSC2 716 SANGER
SU11274 MET RTK signaling GDSC1 918 MGH
Savolitinib AZD6094, Volitinib, AZD-6094, AZD 6094 MET RTK signaling 68289010 GDSC2 957 SANGER
Selumetinib AZD6244, AZD-6244, ARRY-886 MEK1, MEK2 ERK MAPK signaling 10127622 GDSC1 880 SANGER
Selumetinib AZD6244, AZD-6244, ARRY-886 MEK1, MEK2 ERK MAPK signaling 10127622 GDSC1 906 SANGER
Selumetinib AZD6244, AZD-6244, ARRY-886 MEK1, MEK2 ERK MAPK signaling 10127622 GDSC2 949 SANGER
Selumetinib SN1103949345, AZD1480 MEK1, MEK2 ERK MAPK signaling GDSC2 717 SANGER
Serdemetan JNJ-26854165 MDM2 p53 pathway 11609586 GDSC1 924 SANGER
Serdemetan JNJ-26854165 MDM2 p53 pathway 11609586 GDSC2 948 SANGER
Trametinib GSK1120212, Mekinist MEK1, MEK2 ERK MAPK signaling 11707110 GDSC1 881 SANGER
Trametinib GSK1120212, Mekinist MEK1, MEK2 ERK MAPK signaling 11707110 GDSC2 966 SANGER
UNC0638 UNC-0638, UNC 0683 G9a and GLP methyltransferases Chromatin histone methylation 46224516 GDSC1 907 MGH
UNC0638 UNC-0638, UNC 0683 G9a and GLP methyltransferases Chromatin histone methylation 46224516 GDSC1 914 SANGER
ZL049 [(diphenyltetramethylcyclopentadienyl)iridium(III)(2-phenylpyridine)(chloride)] Unclassified GDSC1 913 SANGER
Zoledronate Zoledronic acid, Zometa, Reclast Other GDSC2 717 SANGER
alpha-lipoic acid aLA Metabolism Metabolism None GDSC2 735 SANGER
Feature Name Feature Type
MET_mut coding variant

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