Search Results for: pi3

Name Synonyms Targets Target Pathway PubCHEM Datatset Sample size Screening site
AMG-319 AMG319 PI3K (beta sparing) PI3K/MTOR signaling 68947304 GDSC2 950 SANGER
AS605240 KIN001-173, AS-605240 PI3Kgamma PI3K/MTOR signaling 5289247 GDSC1 908 MGH
AZD6482 AZD 6482, AZD-6482, AK-55409 PI3Kbeta PI3K/MTOR signaling 44137675 GDSC1 876 MGH
AZD6482 AZD 6482, AZD-6482, AK-55409 PI3Kbeta PI3K/MTOR signaling 44137675 GDSC2 267 SANGER
AZD8186 SN1028722848 PI3Kbeta, PI3Kdelta PI3K/MTOR signaling GDSC1 915 SANGER
AZD8186 AZD 8186, AZD-8186 PI3Kalpha, PI3Kbeta PI3K/MTOR signaling 52913813 GDSC2 958 SANGER
AZD8835 SN1040214596 PI3Kalpha, PI3Kdelta PI3K/MTOR signaling GDSC1 909 SANGER
Alpelisib BYL719, BYL-719, NVP-BYL719 PI3Kalpha PI3K/MTOR signaling 56649450 GDSC2 965 SANGER
Apitolisib GDC0980 mTOR, PI3K PI3K/MTOR signaling GDSC1 907 MGH
Buparlisib BKM120, NVP-BKM120 PI3Kalpha, PI3Kdelta, PI3Kbeta, PI3Kgamma PI3K/MTOR signaling 66577015, 16654980 GDSC2 958 SANGER
CZC24832 GTPL6653 PI3Kgamma PI3K/MTOR signaling 42623951 GDSC2 894 SANGER
Dactolisib NVP-BEZ235, BEZ235 PI3K (class 1), MTORC1, MTORC2 PI3K/MTOR signaling 11977753 GDSC1 918 SANGER
Dactolisib NVP-BEZ235, BEZ235 PI3K (class 1), MTORC1, MTORC2 PI3K/MTOR signaling 11977753 GDSC2 958 SANGER
GNE-317 GNE317, GNE 317 PI3Kalpha PI3K/MTOR signaling 70676303 GDSC2 944 SANGER
GSK1059615 PI3K PI3K/MTOR signaling GDSC1 904 MGH
IC-87114 PI3Kdelta PI3K/MTOR signaling GDSC1 913 MGH
Idelalisib CAL-101, Zydelig PI3Kdelta PI3K/MTOR signaling 11625818 GDSC1 914 MGH
Omipalisib GSK2126458, GSK-2126458, EX-8678, GSK458 PI3K (class 1), MTORC1, MTORC2 PI3K/MTOR signaling 25167777 GDSC1 914 MGH
PI-103 PI-103, PI103, PI 103 PI3Kalpha, DAPK3, CLK4, PIM3, HIPK2 Other, kinases 9884685 GDSC1 902 MGH
PI3Ka_4409 SN1037097676 PI3Kalpha, PI3Kdelta PI3K/MTOR signaling GDSC1 913 SANGER
Pictilisib GDC-0941, GDC0941, RG-7621 PI3K (class 1) PI3K/MTOR signaling 17755052 GDSC1 920 SANGER
Pictilisib GDC-0941, GDC0941, RG-7621 PI3K (class 1) PI3K/MTOR signaling 17755052 GDSC1 868 SANGER
Pictilisib GDC-0941, GDC0941, RG-7621 PI3K (class 1) PI3K/MTOR signaling 17755052 GDSC2 967 SANGER
Pilaralisib XL-147 PI3K PI3K/MTOR signaling GDSC1 919 MGH
TGX221 TGX-221, Tgx 221 PI3Kbeta PI3K/MTOR signaling 9907093 GDSC1 398 MGH
Taselisib GDC-0032, GDC0032, RG7604 PI3K (beta sparing) PI3K/MTOR signaling 51001932 GDSC2 966 SANGER
Voxtalisib XL-765, SAR245409 PI3K (class 1), DNAPK, MTOR PI3K/MTOR signaling GDSC1 919 MGH
ZSTK474 KIN001-167, ZSTK-474, ZSTK 474 PI3K (class 1) PI3K/MTOR signaling 11647372 GDSC1 911 MGH

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