Name | Synonyms | Targets | Target Pathway | PubCHEM | Datatset | Sample size | Screening site |
---|---|---|---|---|---|---|---|
AMG-319 | AMG319 | PI3K (beta sparing) | PI3K/MTOR signaling | 68947304 | GDSC2 | 950 | SANGER |
AS605240 | KIN001-173, AS-605240 | PI3Kgamma | PI3K/MTOR signaling | 5289247 | GDSC1 | 908 | MGH |
AZD6482 | AZD 6482, AZD-6482, AK-55409 | PI3Kbeta | PI3K/MTOR signaling | 44137675 | GDSC1 | 876 | MGH |
AZD6482 | AZD 6482, AZD-6482, AK-55409 | PI3Kbeta | PI3K/MTOR signaling | 44137675 | GDSC2 | 267 | SANGER |
AZD8186 | SN1028722848 | PI3Kbeta, PI3Kdelta | PI3K/MTOR signaling | GDSC1 | 915 | SANGER | |
AZD8186 | AZD 8186, AZD-8186 | PI3Kalpha, PI3Kbeta | PI3K/MTOR signaling | 52913813 | GDSC2 | 958 | SANGER |
AZD8835 | SN1040214596 | PI3Kalpha, PI3Kdelta | PI3K/MTOR signaling | GDSC1 | 909 | SANGER | |
Alpelisib | BYL719, BYL-719, NVP-BYL719 | PI3Kalpha | PI3K/MTOR signaling | 56649450 | GDSC2 | 965 | SANGER |
Apitolisib | GDC0980 | mTOR, PI3K | PI3K/MTOR signaling | GDSC1 | 907 | MGH | |
Buparlisib | BKM120, NVP-BKM120 | PI3Kalpha, PI3Kdelta, PI3Kbeta, PI3Kgamma | PI3K/MTOR signaling | 66577015, 16654980 | GDSC2 | 958 | SANGER |
CZC24832 | GTPL6653 | PI3Kgamma | PI3K/MTOR signaling | 42623951 | GDSC2 | 894 | SANGER |
Dactolisib | NVP-BEZ235, BEZ235 | PI3K (class 1), MTORC1, MTORC2 | PI3K/MTOR signaling | 11977753 | GDSC1 | 918 | SANGER |
Dactolisib | NVP-BEZ235, BEZ235 | PI3K (class 1), MTORC1, MTORC2 | PI3K/MTOR signaling | 11977753 | GDSC2 | 958 | SANGER |
GNE-317 | GNE317, GNE 317 | PI3Kalpha | PI3K/MTOR signaling | 70676303 | GDSC2 | 944 | SANGER |
GSK1059615 | PI3K | PI3K/MTOR signaling | GDSC1 | 904 | MGH | ||
IC-87114 | PI3Kdelta | PI3K/MTOR signaling | GDSC1 | 913 | MGH | ||
Idelalisib | CAL-101, Zydelig | PI3Kdelta | PI3K/MTOR signaling | 11625818 | GDSC1 | 914 | MGH |
Omipalisib | GSK2126458, GSK-2126458, EX-8678, GSK458 | PI3K (class 1), MTORC1, MTORC2 | PI3K/MTOR signaling | 25167777 | GDSC1 | 914 | MGH |
PI-103 | PI-103, PI103, PI 103 | PI3Kalpha, DAPK3, CLK4, PIM3, HIPK2 | Other, kinases | 9884685 | GDSC1 | 902 | MGH |
PI3Ka_4409 | SN1037097676 | PI3Kalpha, PI3Kdelta | PI3K/MTOR signaling | GDSC1 | 913 | SANGER | |
Pictilisib | GDC-0941, GDC0941, RG-7621 | PI3K (class 1) | PI3K/MTOR signaling | 17755052 | GDSC1 | 920 | SANGER |
Pictilisib | GDC-0941, GDC0941, RG-7621 | PI3K (class 1) | PI3K/MTOR signaling | 17755052 | GDSC1 | 868 | SANGER |
Pictilisib | GDC-0941, GDC0941, RG-7621 | PI3K (class 1) | PI3K/MTOR signaling | 17755052 | GDSC2 | 967 | SANGER |
Pilaralisib | XL-147 | PI3K | PI3K/MTOR signaling | GDSC1 | 919 | MGH | |
TGX221 | TGX-221, Tgx 221 | PI3Kbeta | PI3K/MTOR signaling | 9907093 | GDSC1 | 398 | MGH |
Taselisib | GDC-0032, GDC0032, RG7604 | PI3K (beta sparing) | PI3K/MTOR signaling | 51001932 | GDSC2 | 966 | SANGER |
Voxtalisib | XL-765, SAR245409 | PI3K (class 1), DNAPK, MTOR | PI3K/MTOR signaling | GDSC1 | 919 | MGH | |
ZSTK474 | KIN001-167, ZSTK-474, ZSTK 474 | PI3K (class 1) | PI3K/MTOR signaling | 11647372 | GDSC1 | 911 | MGH |
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