| AST-1306 |  | EGFR, ERBB4 | RTK signaling |  | GDSC1 | 903 | MGH | 
           | AZD3759 |  | EGFR | EGFR signaling | 78209992 | GDSC2 | 966 | SANGER | 
           | AZD8931 | SN0216062465 | EGFR, ERBB2, ERBB3 | RTK signaling |  | GDSC1 | 913 | SANGER | 
           | Afatinib | BIBW2992, Tovok, Gilotrif | EGFR, ERBB2 | EGFR signaling | 10184653 | GDSC1 | 929 | SANGER | 
           | Afatinib | BIBW2992, Tovok, Gilotrif | EGFR, ERBB2 | EGFR signaling | 10184653 | GDSC1 | 903 | SANGER | 
           | Afatinib | BIBW2992, Tovok, Gilotrif | EGFR, ERBB2 | EGFR signaling | 10184653 | GDSC2 | 966 | SANGER | 
           | Axitinib | AG-13736, Inlyta | PDGFR, KIT, VEGFR | RTK signaling | 6450551 | GDSC1 | 927 | SANGER | 
           | Axitinib | AG-13736, Inlyta | PDGFR, KIT, VEGFR | RTK signaling | 6450551 | GDSC2 | 961 | SANGER | 
           | BIBF-1120 |  | VEGFR, PDGFR, FGFR | RTK signaling |  | GDSC1 | 918 | MGH | 
           | Brivanib, BMS-540215 |  | VEGFR, PDGFR | RTK signaling |  | GDSC1 | 918 | MGH | 
           | CI-1033 |  | EGFR, ERBB2, ERBB4 | RTK signaling |  | GDSC1 | 916 | MGH | 
           | CUDC-101 | CUDC 101 | HDAC1-10, EGFR, ERBB2 | Other | 24756910 | GDSC1 | 893 | MGH | 
           | Cabozantinib | BMS-907351, XL-184, Cometriq | VEGFR, MET, RET, KIT, FLT1, FLT3, FLT4, TIE2,AXL | RTK signaling | 25102847 | GDSC1 | 911 | MGH | 
           | Cediranib | AZD2171, AZD 2171, AZD-2171, Recentin | VEGFR, FLT1, FLT2, FLT3, FLT4, KIT, PDGFRB | RTK signaling | 9933475 | GDSC2 | 958 | SANGER | 
           | Cetuximab | Erbitux, IMC-C225, C225, IMC-225, L01XC06 | EGFR | EGFR signaling | 85668777 | GDSC1 | 862 | SANGER | 
           | Erlotinib | Tarceva, RG-1415, CP-358774, OSI-774, Ro-508231, R-1415 | EGFR | EGFR signaling | 176870 | GDSC1 | 393 | MGH | 
           | Erlotinib | Tarceva, RG-1415, CP-358774, OSI-774, Ro-508231, R-1415 | EGFR | EGFR signaling | 176870 | GDSC2 | 955 | SANGER | 
           | Foretinib | GSK1363089, XL-880, EXEL-2880, GSK089 | MET, KDR, TIE2, VEGFR3/FLT4, RON, PDGFR, FGFR1, EGFR | RTK signaling | 42642645 | GDSC1 | 909 | MGH | 
           | Foretinib | GSK1363089, XL-880, EXEL-2880, GSK089 | MET, KDR, TIE2, VEGFR3/FLT4, RON, PDGFR, FGFR1, EGFR | RTK signaling | 42642645 | GDSC2 | 953 | SANGER | 
           | Gefitinib | ZD-1839, Iressa | EGFR | EGFR signaling | 123631 | GDSC1 | 927 | SANGER | 
           | Gefitinib | ZD-1839, Iressa | EGFR | EGFR signaling | 123631 | GDSC2 | 958 | SANGER | 
           | Lapatinib | Tykerb, Tyverb | EGFR, ERBB2 | RTK signaling | 208908 | GDSC1 | 395 | MGH | 
           | Lapatinib | Tykerb, Tyverb | EGFR, ERBB2 | EGFR signaling | 208908 | GDSC2 | 966 | SANGER | 
           | Linifanib | ABT-869, ABT 869 | VEGFR1, VEGFR2, VEGFR3, CSF1R, FLT3, KIT | RTK signaling | 11485656 | GDSC1 | 914 | MGH | 
           | Motesanib | AMG-706, AMG 706, AMG706 | VEGFR, RET, KIT, PDGFR | RTK signaling | 11667893 | GDSC1 | 927 | SANGER | 
           | Motesanib | AMG-706, AMG 706, AMG706 | VEGFR, RET, KIT, PDGFR | RTK signaling | 11667893 | GDSC2 | 949 | SANGER | 
           | OSI-930 | OSI 930 OSI930 | KIT, VEGFR2 | RTK signaling | 9868037 | GDSC1 | 913 | MGH | 
           | Osimertinib | AZD9291, AZD 9291, AZD-9291, Tagrisso, Mereletinib | EGFR | EGFR signaling | 71496458 | GDSC2 | 957 | SANGER | 
           | PF-00299804 |  | EGFR, ERBB2, ERBB4 | RTK signaling |  | GDSC1 | 909 | MGH | 
           | Pelitinib | EKB-569, EKB 569 | EGFR | EGFR signaling | 6445562 | GDSC1 | 913 | MGH | 
           | Ponatinib | AP24534, AP-24534, KIN001-192, Iclusig | ABL, PDGFRA, VEGFR2, FGFR1, SRC, TIE2, FLT3 | Other, kinases | 24826799 | GDSC1 | 877 | MGH | 
           | Sapitinib | AZD8931 | EGFR, ERBB2, ERBB3 | EGFR signaling | 11488320 | GDSC2 | 966 | SANGER | 
           | Sorafenib | Nexavar, 284461-73-0, BAY 43-9006 | PDGFR, KIT, VEGFR, RAF | RTK signaling | 216239 | GDSC1 | 396 | MGH | 
           | Sorafenib | Nexavar, 284461-73-0, BAY 43-9006 | PDGFR, KIT, VEGFR, RAF | Other, kinases | 216239 | GDSC2 | 958 | SANGER | 
           | Sunitinib | Sutent, Sunitinib Malate, SU-11248 | PDGFR, KIT, VEGFR, FLT3, RET, CSF1R | RTK signaling | 5329102 | GDSC1 | 396 | MGH | 
           | Tivozanib | AV-951, AV 951, KRN-951, KIL8951, ASP-4130 | VEGFR1, VEGFR2, VEGFR3, PDGFR, KIT | RTK signaling | 9911830 | GDSC1 | 912 | MGH |