Name | Synonyms | Targets | Target Pathway | PubCHEM | Datatset | Sample size | Screening site |
---|---|---|---|---|---|---|---|
Cabozantinib | BMS-907351, XL-184, Cometriq | VEGFR, MET, RET, KIT, FLT1, FLT3, FLT4, TIE2,AXL | RTK signaling | 25102847 | GDSC1 | 911 | MGH |
Cediranib | AZD2171, AZD 2171, AZD-2171, Recentin | VEGFR, FLT1, FLT2, FLT3, FLT4, KIT, PDGFRB | RTK signaling | 9933475 | GDSC2 | 958 | SANGER |
Midostaurin | PKC412, benzoylstaurosporine, CGP-41251 | PKC, PPK, FLT1, c-FGR, others | Other | several | GDSC1 | 881 | MGH |
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