Name | Synonyms | Targets | Target Pathway | PubCHEM | Datatset | Sample size | Screening site |
---|---|---|---|---|---|---|---|
BMS-536924 | BMS 536924 | IGF1R, IR | IGF1R signaling | 10390396 | GDSC1 | 396 | MGH |
BMS-536924 | BMS 536924 | IGF1R, IR | IGF1R signaling | 10390396 | GDSC1 | 909 | SANGER |
BMS-536924 | BMS 536924 | IGF1R, IR | IGF1R signaling | 10390396 | GDSC2 | 958 | SANGER |
BMS-754807 | BMS754807, BMS 754807 | IGF1R, IR | RTK signaling | 24785538 | GDSC1 | 865 | MGH |
BMS-754807 | BMS-754807 | IGF1R, IR | IGF1R signaling | GDSC2 | 949 | SANGER | |
GSK1904529A | GSK-1904529A, GSK 1904529A | IGF1R, IR | RTK signaling | 25124816 | GDSC1 | 870 | MGH |
GSK1904529A | GSK-1904529A, GSK 1904529A | IGF1R, IR | IGF1R signaling | 25124816 | GDSC2 | 965 | SANGER |
IGF1R_3801 | SN1051640224, IGF1R_3801 | IGFR1 | IGF1R signaling | GDSC2 | 716 | SANGER | |
IGFR_3801 | SN1056768819 | IGFR1 | IGF1R signaling | GDSC1 | 915 | SANGER | |
Idelalisib | CAL-101, Zydelig | PI3Kdelta | PI3K/MTOR signaling | 11625818 | GDSC1 | 914 | MGH |
Linsitinib | OSI-906, ASP-7487 | IGF1R | IGF1R signaling | 11640390 | GDSC1 | 867 | MGH |
Linsitinib | OSI-906, ASP-7487 | IGF1R | IGF1R signaling | 11640390 | GDSC2 | 966 | SANGER |
NVP-ADW742 | NVP ADW742, NVPADW742 | IGF1R | IGF1R signaling | 9825149 | GDSC2 | 958 | SANGER |
Nilotinib | Tasigna, AMN 107 | ABL | ABL signaling | 644241 | GDSC1 | 933 | SANGER |
Nilotinib | Tasigna, AMN 107 | ABL | ABL signaling | 644241 | GDSC2 | 955 | SANGER |
Phenformin | DBI | Biguanide agent | Other | 8249 | GDSC1 | 901 | MGH |
Ponatinib | AP24534, AP-24534, KIN001-192, Iclusig | ABL, PDGFRA, VEGFR2, FGFR1, SRC, TIE2, FLT3 | Other, kinases | 24826799 | GDSC1 | 877 | MGH |
Thapsigargin | Octanoic acid | SERCA | Other | 446378 | GDSC1 | 852 | MGH |
glutathione | G6013, sigma | anti-oxidant proteins | Other | GDSC2 | 732 | SANGER |
Name | Cell Model Passport Link | COSMIC ID | Tissue | Tissue sub-type |
---|---|---|---|---|
IGR-1 | SIDM01060 | 907169 | SKCM | Skin |
IGR-1 | SIDM01060 | 907169 | SKCM | Skin |
IGR-37 | SIDM01066 | 1240153 | SKCM | Skin |
IGR-37 | SIDM01066 | 1240153 | SKCM | Skin |
IGROV-1 | SIDM00151 | 905968 | OV | Urogenital system |
IGROV-1 | SIDM00151 | 905968 | OV | Urogenital system |
SIG-M5 | SIDM00396 | 909715 | LAML | Blood |
SIG-M5 | SIDM00396 | 909715 | LAML | Blood |
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