Name | Synonyms | Targets | Target Pathway | PubCHEM | Datatset | Sample size | Screening site |
---|---|---|---|---|---|---|---|
AZ960 | AZ 960, AZ-960 | JAK2, JAK3 | Other, kinases | 25099184 | GDSC2 | 892 | SANGER |
AZD1480 | SN1044232195 | JAK1, JAK2 | Other, kinases | GDSC1 | 921 | SANGER | |
Fedratinib | TG101348, TG-101348, SAR302503, SAR-302503 | JAK2 | Other, kinases | 16722836 | GDSC1 | 914 | MGH |
GSK2276186C | JAK1, JAK2, JAK3 | Other, kinases | GDSC2 | 717 | SANGER | ||
JAK_8517 | SN1066590414, JAK_8517 | JAK1, JAK2 | Other, kinases | GDSC2 | 717 | SANGER | |
Lestaurtinib | CEP-701, SP-924, SPM-924, A-154475, KT-555 | FLT3, JAK2, NTRK1, NTRK2, NTRK3 | Other, kinases | 126565 | GDSC1 | 929 | SANGER |
Lestaurtinib | CEP-701, SP-924, SPM-924, A-154475, KT-555 | FLT3, JAK2, NTRK1, NTRK2, NTRK3 | Other, kinases | 126565 | GDSC2 | 947 | SANGER |
Ruxolitinib | INCB-18424, Ruxolitinib Phosphate, Jakafi | JAK1, JAK2 | Other, kinases | 25126798 | GDSC1 | 916 | MGH |
Ruxolitinib | INCB-18424, Ruxolitinib Phosphate, Jakafi | JAK1, JAK2 | Other, kinases | 25126798 | GDSC2 | 898 | SANGER |
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