Name | Synonyms | Targets | Target Pathway | PubCHEM | Datatset | Sample size | Screening site |
---|---|---|---|---|---|---|---|
Amuvatinib | MP470, MP 470, MP-470 | KIT, PDGFRA, FLT3 | RTK signaling | 11282283 | GDSC1 | 906 | MGH |
Masitinib | AB1010, Masivet | KIT, PDGFRA, PDGFRB | RTK signaling | 10074640 | GDSC1 | 913 | MGH |
Pazopanib | Votrient | CSF1R, KIT, PDGFRA, PDGFRB | RTK signaling | 10113978 | GDSC1 | 866 | MGH |
Ponatinib | AP24534, AP-24534, KIN001-192, Iclusig | ABL, PDGFRA, VEGFR2, FGFR1, SRC, TIE2, FLT3 | Other, kinases | 24826799 | GDSC1 | 877 | MGH |
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