Search Results for: t3

Name Synonyms Targets Target Pathway PubCHEM Datatset Sample size Screening site
A-443654 KIN001-139 AKT1, AKT2, AKT3 PI3K/MTOR signaling 10172943 GDSC1 397 MGH
AKT inhibitor VIII Akti-1/2, KIN001-102 AKT1, AKT2, AKT3 PI3K/MTOR signaling 10196499 GDSC1 877 MGH
AKT inhibitor VIII Akti-1/2, KIN001-102 AKT1, AKT2, AKT3 PI3K/MTOR signaling 10196499 GDSC1 913 MGH
AZD5363 AKT1, AKT2, AKT3, ROCK2 Other, kinases 25227436, 42602260 GDSC2 958 SANGER
Afuresertib GSK2110183, GSK2110183C AKT1, AKT2, AKT3 PI3K/MTOR signaling 46843057 GDSC2 957 SANGER
Amuvatinib MP470, MP 470, MP-470 KIT, PDGFRA, FLT3 RTK signaling 11282283 GDSC1 906 MGH
BAY AKT1 AKT1, AKT2, AKT3 Apoptosis regulation GDSC1 835 SANGER
Cabozantinib BMS-907351, XL-184, Cometriq VEGFR, MET, RET, KIT, FLT1, FLT3, FLT4, TIE2,AXL RTK signaling 25102847 GDSC1 911 MGH
Cediranib AZD2171, AZD 2171, AZD-2171, Recentin VEGFR, FLT1, FLT2, FLT3, FLT4, KIT, PDGFRB RTK signaling 9933475 GDSC2 958 SANGER
GSK2110183B AKT1, AKT2, AKT3 PI3K/MTOR signaling GDSC2 717 SANGER
GSK690693 GSK 690693, GSK-690693 AKT1, AKT2, AKT3 PI3K/MTOR signaling 16725726 GDSC1 910 MGH
Ipatasertib GDC0068, GDC 0068, GDC-0068 AKT1, AKT, AKT3 PI3K/MTOR signaling 24788740 GDSC2 958 SANGER
Lestaurtinib CEP-701, SP-924, SPM-924, A-154475, KT-555 FLT3, JAK2, NTRK1, NTRK2, NTRK3 Other, kinases 126565 GDSC1 929 SANGER
Lestaurtinib CEP-701, SP-924, SPM-924, A-154475, KT-555 FLT3, JAK2, NTRK1, NTRK2, NTRK3 Other, kinases 126565 GDSC2 947 SANGER
Linifanib ABT-869, ABT 869 VEGFR1, VEGFR2, VEGFR3, CSF1R, FLT3, KIT RTK signaling 11485656 GDSC1 914 MGH
Ponatinib AP24534, AP-24534, KIN001-192, Iclusig ABL, PDGFRA, VEGFR2, FGFR1, SRC, TIE2, FLT3 Other, kinases 24826799 GDSC1 877 MGH
Quizartinib AC220, AC 220, AC-220, Asp-2689 FLT3 RTK signaling 24889392 GDSC1 914 MGH
Sunitinib Sutent, Sunitinib Malate, SU-11248 PDGFR, KIT, VEGFR, FLT3, RET, CSF1R RTK signaling 5329102 GDSC1 396 MGH
Telomerase Inhibitor IX MST-312, MST 312, MST312 Telomerase Genome integrity 10385095 GDSC2 958 SANGER
Uprosertib GSK2141795, GSK2141795C, GSK-2141795 AKT1, AKT2, AKT3 PI3K/MTOR signaling 51042438 GDSC2 898 SANGER
Uprosertib GSK2141795, GSK2141795C, GSK-2141795 AKT1, AKT2, AKT3 PI3K/MTOR signaling 51042438 GDSC2 736 SANGER
WZ3105 SRC, ROCK2, NTRK2, FLT3, IRAK1, others Other none GDSC1 914 MGH
Name Cell Model Passport Link COSMIC ID Tissue Tissue sub-type
HuP-T3 SIDM00533 907285 PAAD Pancreas
HuP-T3 SIDM00533 907285 PAAD Pancreas
Feature Name Feature Type
CNOT3_mut coding variant
DNMT3A_mut coding variant
FLT3_mut coding variant

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