Search Results for: th

Name Synonyms Targets Target Pathway PubCHEM Datatset Sample size Screening site
5-azacytidine DNA methyltransferases Other GDSC2 740 SANGER
BDILV000379a 4-(4-(1-methyl-1H-pyrazol-4-yl)-1-(2-(1-methyl-1H-pyrazol-4-yl)ethyl)-4,5-dihydro-1H-imidazol-5-yl)benzonitrile BAZ2A, BAZ2B Chromatin histone acetylation GDSC2 717 SANGER
BDOCA000347a 4-bromo-N-(6-methoxy-1,3-dimethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)-2-methylbenzenesulfonamide BRPF1, BRPF2, BRPF3 Chromatin histone acetylation GDSC2 717 SANGER
Bromosporine ethyl N-[6-(3-methanesulfonamido-4-methylphenyl)-3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-8-yl]carbamate CECR2, BRD2, BRD4, BRD9 Chromatin other GDSC2 716 SANGER
Camptothecin Camptothecine, (+)-Camptothecin TOP1 DNA replication 24360 GDSC2 968 SANGER
DMOG Dimethyloxalylglcine HIF-PH Metabolism 560326 GDSC1 876 MGH
Doxorubicin Doxil, Rubex, Adriamycin, Adriablastin, Doxorubicine Anthracycline DNA replication 31703 GDSC1 870 MGH
Doxorubicin Anthracycline DNA replication GDSC1 922 SANGER
Epirubicin Ellence, Farmorubicin, IMI-28 Anthracycline DNA replication 41867 GDSC2 958 SANGER
Epothilone B Patupilone, EpoB, EPO906, GNF-PF-193 Microtubule stabiliser Mitosis 448013 GDSC1 868 MGH
FY026 [(para-cymene)osmium(N,N-dimethylphenlyazopyridine)(iodide)]hexafluorophophate Unclassified GDSC1 915 SANGER
GSK2801 1-(7-(2-methylsulfonyl-phenyl)-4-propoxy-1-aza-bicyclo[4.3.0]nona-2,4,6,8-tetraen-9-yl)-ethanone Chromatin other GDSC2 717 SANGER
Leflunomide Sulol, SU-101, HWA-486, Arava Pyrimidine synthesis inhibitor DNA replication 3899 GDSC2 894 SANGER
Methotrexate Abitrexate, Amethopterin, Rheumatrex, Trexall, Folex Antimetabolite DNA replication 126941 GDSC1 933 SANGER
Methotrexate Abitrexate, Amethopterin, Rheumatrex, Trexall, Folex Antimetabolite DNA replication 126941 GDSC2 881 SANGER
Midostaurin PKC412, benzoylstaurosporine, CGP-41251 PKC, PPK, FLT1, c-FGR, others Other several GDSC1 881 MGH
N23918-95-7 JMJ histone demethylase Chromatin histone methylation GDSC1 913 SANGER
N24798-49-A1 JMJ histone demethylase Chromatin histone methylation GDSC1 908 SANGER
Parthenolide HDAC1 Chromatin histone acetylation 7251185 GDSC1 400 MGH
Pyrimethamine Daraprim, Chloridine Dihydrofolate reductase (DHFR) Other 4993 GDSC1 398 MGH
SGC-CBP30 8-(3-chloro-4-methoxy-phenethyl)-4-(3,5-dimethyl-isoxazol-4-yl)-9-(2-(morpholin-4-yl)-propyl)-7,9-diaza-bicyclo[4.3.0]nona-1(6),2,4,7-tetraene EP300, CBP Chromatin histone acetylation GDSC2 716 SANGER
SN-38 7-Ethyl-10-Hydroxy-Camptothecin, SN 38 TOP1 DNA replication 104842 GDSC1 938 SANGER
SN-38 7-Ethyl-10-Hydroxy-Camptothecin, SN 38 TOP1 DNA replication 104842 GDSC2 958 SANGER
Schweinfurthin A Unclassified GDSC2 716 SANGER
THR-101 WIMM synthesis Mutant RAS PI3K/MTOR signaling None GDSC2 731 SANGER
THR-102 WIMM synthesis Mutant RAS PI3K/MTOR signaling None GDSC2 731 SANGER
THR-103 WIMM synthesis Mutant RAS PI3K/MTOR signaling None GDSC2 731 SANGER
THZ-1-87 BTK, BMX Other, kinases GDSC1 99 SANGER
THZ-2-102-1 CDK7 Cell cycle none GDSC1 890 MGH
THZ-2-49 CDK9 Cell cycle none GDSC1 899 MGH
THZ-2-98-01 IRAK1 Unclassified GDSC1 99 SANGER
Thapsigargin Octanoic acid SERCA Other 446378 GDSC1 852 MGH
Tozasertib MK 0457,MK-0457,MK-045, VX-680 VX 680 VX-68 AURKA, AURKB, AURKC, others Mitosis 5494449 GDSC1 392 MGH
Tozasertib MK 0457,MK-0457,MK-045, VX-680 VX 680 VX-68 AURKA, AURKB, AURKC, others Mitosis 5494449 GDSC2 268 SANGER
UNC0638 UNC-0638, UNC 0683 G9a and GLP methyltransferases Chromatin histone methylation 46224516 GDSC1 907 MGH
UNC0638 UNC-0638, UNC 0683 G9a and GLP methyltransferases Chromatin histone methylation 46224516 GDSC1 914 SANGER
WZ3105 SRC, ROCK2, NTRK2, FLT3, IRAK1, others Other none GDSC1 914 MGH
XMD14-99 ALK, CDK7, LTK, others Other, kinases none GDSC1 914 MGH
ZL049 [(diphenyltetramethylcyclopentadienyl)iridium(III)(2-phenylpyridine)(chloride)] Unclassified GDSC1 913 SANGER
Zibotentan ZD4054, ZD-4054 Endothelin-1 receptor (EDNRA) Other 9910224 GDSC1 912 MGH
glutathione G6013, sigma anti-oxidant proteins Other GDSC2 732 SANGER
Name Cell Model Passport Link COSMIC ID Tissue Tissue sub-type
CGTH-W-1 SIDM01248 910568 THCA Thyroid
CGTH-W-1 SIDM01248 910568 THCA Thyroid
THP-1 SIDM01172 909771 LAML Blood
THP-1 SIDM01172 909771 LAML Blood
Feature Name Feature Type
THRAP3_mut coding variant

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