association id |
FEATURE |
Drug id |
Propr |
Public |
Drug Name |
Drug Target |
N FEATURE pos |
N FEATURE neg |
log max Conc tested |
FEATURE neg logIC50 MEAN |
FEATURE pos logIC50 MEAN |
FEATURE deltaMEAN IC50 |
FEATURE IC50 effectSize |
FEATURE neg Glass delta |
FEATURE pos Glass delta |
ANOVA FEATURE pval |
Tissue ANOVA pval |
MSI ANOVA pval |
ANOVA FEATURE FDR % |
a161 |
gain_cnaPANCAN363_(ASXL1) |
1017 |
1 |
1 |
Olaparib |
PARP1, PARP2 |
85 |
762 |
1.61 |
3.47 |
4.09 |
0.615 |
0.61 . |
0.59 . |
0.78 . |
5.05e-05 |
8.14e-21 |
2.23e-01 |
5.2 |
a195 |
gain_cnaPANCAN363_(ASXL1) |
1529 |
1 |
1 |
MLN4924 |
NEDD8-activating enzyme |
76 |
626 |
0 |
0.13 |
0.896 |
0.766 |
0.51 . |
0.51 . |
0.48 |
7.82e-05 |
1.04e-07 |
4.8e-02 |
6.6 |
a219 |
gain_cnaPANCAN363_(ASXL1) |
1018 |
1 |
1 |
ABT-888 |
PARP1, PARP2 |
84 |
763 |
1.61 |
3.87 |
4.29 |
0.424 |
0.6 . |
0.59 . |
0.66 . |
1.06e-04 |
8.57e-19 |
2.35e-01 |
7.9 |
a267 |
gain_cnaPANCAN363_(ASXL1) |
1378 |
1 |
1 |
Bleomycin (50 uM) |
DNA damage |
101 |
831 |
3.91 |
2.26 |
2.87 |
0.609 |
0.29 |
0.29 |
0.31 |
1.79e-04 |
6.04e-31 |
3.34e-04 |
11 |
a276 |
gain_cnaPANCAN363_(ASXL1) |
1003 |
1 |
1 |
Camptothecin |
TOP1 |
85 |
761 |
-2.3 |
-4.14 |
-3.18 |
0.959 |
0.54 . |
0.54 . |
0.54 . |
1.93e-04 |
2.88e-23 |
1.05e-01 |
12 |
a288 |
gain_cnaPANCAN363_(ASXL1) |
208 |
1 |
1 |
SB-715992 |
KIF11 |
102 |
820 |
-2.06 |
-1.87 |
-1.01 |
0.861 |
0.49 |
0.48 |
0.52 . |
2.13e-04 |
1.92e-33 |
1.9e-02 |
12 |
a333 |
gain_cnaPANCAN363_(ASXL1) |
1495 |
1 |
1 |
AZD-2281 |
PARP1, PARP2 |
97 |
806 |
2.3 |
3.57 |
4 |
0.432 |
0.42 |
0.41 |
0.43 |
3.01e-04 |
8.5e-17 |
1.39e-03 |
15 |
a365 |
gain_cnaPANCAN363_(ASXL1) |
300 |
1 |
1 |
CX-5461 |
RNA Pol I |
99 |
818 |
2.33 |
2.88 |
3.95 |
1.07 |
0.54 . |
0.53 . |
0.66 . |
3.69e-04 |
8.82e-45 |
2.24e-01 |
17 |
a386 |
gain_cnaPANCAN363_(ASXL1) |
1239 |
1 |
1 |
YK 4-279 |
RNA helicase A |
82 |
710 |
2.3 |
1.5 |
2.02 |
0.523 |
0.41 |
0.42 |
0.38 |
4.14e-04 |
1.4e-08 |
4.47e-02 |
18 |
a414 |
gain_cnaPANCAN363_(ASXL1) |
179 |
1 |
1 |
5-Fluorouracil |
DNA antimetabolite |
99 |
814 |
3.47 |
3.47 |
4.35 |
0.884 |
0.5 . |
0.49 |
0.6 . |
5.01e-04 |
2.51e-45 |
2.32e-01 |
20 |
a441 |
gain_cnaPANCAN363_(ASXL1) |
266 |
1 |
1 |
Zibotentan, ZD4054 |
Endothelin A Receptor |
101 |
818 |
3 |
5.45 |
5.74 |
0.289 |
0.51 . |
0.51 . |
0.61 . |
5.57e-04 |
1.73e-49 |
1.87e-01 |
21 |
a485 |
gain_cnaPANCAN363_(ASXL1) |
1005 |
1 |
1 |
Cisplatin |
DNA crosslinker |
85 |
762 |
1.79, 2.30 |
2.83 |
3.39 |
0.556 |
0.47 |
0.46 |
0.5 . |
6.71e-04 |
4.6e-17 |
5.52e-01 |
23 |